Proparacaine hydrochloride

CAS No. 5875-06-9

Proparacaine hydrochloride ( Proxymetacaine hydrochloride )

Catalog No. M15166 CAS No. 5875-06-9

An irreversible local anesthetic; inhibits pain sensations that is believed to act as an antagonist on voltage-gated sodium channels.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
50MG 32 In Stock
100MG 45 In Stock
200MG 65 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Proparacaine hydrochloride
  • Note
    Research use only, not for human use.
  • Brief Description
    An irreversible local anesthetic; inhibits pain sensations that is believed to act as an antagonist on voltage-gated sodium channels.
  • Description
    An irreversible local anesthetic; inhibits pain sensations that is believed to act as an antagonist on voltage-gated sodium channels.Pain Approved
  • Synonyms
    Proxymetacaine hydrochloride
  • Pathway
    Membrane Transporter/Ion Channel
  • Target
    Sodium Channel
  • Recptor
    Voltage-gatedsodiumchannel
  • Research Area
    Neurological Disease
  • Indication
    Pain

Chemical Information

  • CAS Number
    5875-06-9
  • Formula Weight
    330.85
  • Molecular Formula
    C16H27ClN2O3
  • Purity
    >98% (HPLC)
  • Solubility
    10 mM in DMSO
  • SMILES
    CCCOC1=C(C=C(C=C1)C(=O)OCCN(CC)CC)N.Cl
  • Chemical Name
    Benzoic acid, 3-amino-4-propoxy-, 2-(diethylamino)ethyl ester, hydrochloride (1:1)

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Gusovsky F, et al. Brain Res. 1990 Jun 4;518(1-2):101-6.
2. McAlvin JB, et al. Invest Ophthalmol Vis Sci. 2015 Jun;56(6):3820-6.
3. Hung CH, et al. Anesth Analg. 2010 Jan 1;110(1):238-42.
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